Efficient and convenient preparation of 3-aryl-2,2-dimethylpropanoates via Negishi coupling.

نویسندگان

  • Young-Shin Kwak
  • Aaron D Kanter
  • Bing Wang
  • Yugang Liu
چکیده

An efficient and convenient Negishi coupling protocol was developed for the preparation of 3-aryl-2,2-dimethylpropanoates providing easy access to key pharmaceutical intermediates that often require multi-step synthesis using conventional enolate chemistry.

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عنوان ژورنال:
  • Chemical communications

دوره 16  شماره 

صفحات  -

تاریخ انتشار 2009